Description
Buy LY-2183240 for sale
Buy LY-2183240 for sale. LY-2183240 for sale is a drug which acts both as a potent inhibitor of the reuptake of the endocannabinoid anandamide and as an inhibitor of fatty acid amide hydrolase (FAAH), the primary enzyme responsible for degrading anandamide. This leads to markedly elevated anandamide levels in the brain, and Buy LY-2183240 online for sale has been shown to produce both analgesic and anxiolytic effects in animal models. While buy LY-2183240 online is a potent inhibitor of FAAH, it has relatively poor selectivity and also inhibits several other enzyme side targets. Consequently, it was never developed for clinical use, though it remains widely used in research, and has also been sold as a designer drug. LY-2183240 for sale
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Biological Activity for LY 2183240
LY 2183240 for sale is a novel and highly potent blocker of anandamide uptake (IC50 = 270 pM). Inhibits fatty acid amide hydrolase (FAAH) activity (IC50 = 12.4 nM). Following i.p. administration in rats, increases brain anandamide concentration and exerts antinociceptive effects in formalin model of pain.
Licensing Information of LY 2183240 for sale
Sold under license from Eli Lilly and Company
Technical Data for LY 2183240
| M. Wt | 307.35 |
| Formula | C17H17N5O |
| Storage | Store at +4°C |
| Purity | ≥98% (HPLC) |
| CAS Number | 874902-19-9 |
| PubChem ID | 11507802 |
| InChI Key | GZNIYOXWFCDBBJ-UHFFFAOYSA-N |
| Smiles | CN(C)C(=O)N1N=NN=C1CC1=CC=C(C=C1)C1=CC=CC=C1 |
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.
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